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Protein Kinase Information : List of Protein Kinase Inhibitor
# Name of Kinase Name of Inhibitor
1 PKA H-89, HA-1004, H-7, H-8, HA-100, staurosporine
2 PKG H-7, H-8, HA-1004, H-89
3 PKC bisindolylmaleimide IX, chelerythrine, edelfosine, edelfosina, ET18OCH3, H-7, HA-100, H89, HA-1004, Ro 31-8220, staurosporine
4 ABL PP1
5 Adenosine kinase 5-Iodotubercidin
6 Akt/PKB Triciribine (TCN, Tricyclic Nucleoside, NSC-154020, API-2)
7 AMPK indirubin-3'-oxime, 5-Iodotubercidin, H-89
8 BTK  LFM-A13
9 CaMKII KN-62, W-7, HA-1004, HA-1077
10 CDK1, CDK2, CDK5 aloisine, aloisine A, alsterpaullone, indirubin-3'-oxime, kenpaullone, olomoucine, purvalanol A, roscovitine
11 CHK1 H-89
12 CK1  DRB
13 CK2  TBB, DRB
14 EGF-R kinase erbstatin analog, erlotinib, gefitinib, PD 153035, Tyrphostin AG 490, Tyrphostin AG 825, PP1, PP2
15 ERK kinase PD 98059, SL327, olomoucine, 5-Iodotubercidin
16 FYN PP1, PP2, SU6656
17 GSK3 aloisine, aloisine A, indirubin-3'-oxime, kenpaullone
18 HCK PP2
19 HER2 Tyrphostin AG 825
20 IGF1-R PTK inhibitor Tyrphostin AG 1024
21 JAK Tyrphostin AG 490
22 JNK aloisine A, SP600125
23 KIT PP1
24 LCK aminogenistein, PP1, PP2, indirubin-3'-oxime, kenpaullone
25 LYN SU6656
26 MAPKAP-K1b HA-1077
27 MAPK SB202190, SB203580
28 MAPKK arctigenin, PD 98059, SL327, U0126
29 MEK PD 98059, SL327, U0126
30 MKK arctigenin, PD 98059, SL327, U0126
31 MLCK ML-9, W-7, HA-100, HA-1004, H-7, H-8, HA-1077
32 MSK1 H-89, ML-9, HA-1077
33 P38 MAPK SB202190, SB203580
34 PDGF-R kinase DMPQ
35 PI3K LY294002
36 PRK2 HA-1077
37 RHO kinase HA-1077
38 ROCK Y-27632, H-89, ML-9, HA-1077
39 S6K1 rapamycin, sirolimus, H-89, ML-9, HA-1077
40 SAPK PD 169316, SB202190, SB203580
41 SGK indirubin-3'-oxime, H-89
42 SRC familiy PTK PP1, PP2, SU6656
43 SYK piceatannol
44 TOR rapamycin, sirolimus
45 PTK aminogenistein, DMPQ, erbstatin analog, erlotinib, gefitinib, LFM-A13, PD 153035, piceatannol, PP1, PP2, SU 4312, SU6656, Tyrphostin AG 490, Tyrphostin AG 825
46 VEGF-R kinase SU 4312
47 YES SU6656
48 ZAP70 piceatannol